Herpesvirus Antiviral Resistance
Database


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    M460V

    Antiviral assays:

    Antiviral EC50 ratio Phenotype Strain Source Marker Assay Reference
    Filociclovir 4.00 Intermediate level resistance Laboratory strain Recombinant Details Cytomegalovirus UL97 mutations affecting cyclopropavir and ganciclovir susceptibility. (Jan 2011)
    Maribavir 0.30 Possible hypersensitivity, no resistance Laboratory strain Recombinant Details Ganciclovir and maribavir cross-resistance revisited: Relative drug susceptibilities of canonical cytomegalovirus mutants. (Feb 2024)
    Ganciclovir 9.10 High level resistance Recombinant Recombinant Details Ganciclovir and maribavir cross-resistance revisited: Relative drug susceptibilities of canonical cytomegalovirus mutants. (Feb 2024)

    Mutations at the same locus:

    Mutant Resistances
    M460I Filociclovir: High level resistance
    M460I Maribavir: Possible hypersensitivity, no resistance
    M460I Ganciclovir: High level resistance
    M460L
    M460T Ganciclovir: High level resistance